Abstract
α,β-Differentiated 1,2-vicinal diamines have been efficiently synthesized by using new electrophilic imidazolination reaction of alkenes. The hydrolysis of imidazolines was performed by treatment with 6 M HCl in THF at 70°C without epimerization. Eight examples were examined to give good to excellent yields (87-96%).
Original language | English |
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Pages (from-to) | 2919-2921 |
Number of pages | 3 |
Journal | Organic and Biomolecular Chemistry |
Volume | 1 |
Issue number | 16 |
DOIs | |
State | Published - Aug 21 2003 |